Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
P2Y purinoceptor 2
(Homo sapiens (Human))
National Institute Of Diabetes
Curated by
ChEMBL
Ligand
BDBM50422385
(2-Chloro-Adenosinetriphosphate | CHEMBL1368696)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.30E+3nM
Assay Description:
Agonist activity by measuring inositol phosphate accumulation in 1321N1 human astrocytoma cells stably expressing human P2Y purinoceptor 2
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
P2Y purinoceptor 1
(Rattus norvegicus)
Bar-Ilan University
Curated by
ChEMBL
Ligand
BDBM50422406
(2-Chloroadenosine Triphosphate Tetrasodium | CHEMB...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 3.60nM
Assay Description:
Agonists activity was evaluated by release of [Ca2+] release of HEK 293 cells stably transfected with rat-brain P2Y purinoceptor 1 (P2Y1-R)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
P2Y purinoceptor 1
(Homo sapiens (Human))
National Institute Of Diabetes
Curated by
ChEMBL
Ligand
BDBM50422385
(2-Chloro-Adenosinetriphosphate | CHEMBL1368696)
Copy SMILES
Copy InChI
Affinity Data
EC50: 770nM
Assay Description:
Accumulation of inositol phosphate in 1321N1 astrocytoma cells expressing human P2Y1 purinoceptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
P2Y purinoceptor 1
(Meleagris gallopavo)
National Institute Of Diabetes
Curated by
ChEMBL
Ligand
BDBM50422385
(2-Chloro-Adenosinetriphosphate | CHEMBL1368696)
Copy SMILES
Copy InChI
Affinity Data
EC50: 720nM
Assay Description:
Activation of Purinoceptor P2Y1-mediated phospholipase C in turkey erythrocyte membranes
More data for this Ligand-Target Pair
Target Info
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI