Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
Ki: 39.8nMAssay Description:Displacement of [3H]-histamine from human histamine H4 receptor expressed in HEK293 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
Ki: 40nM ΔG°: -42.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
Ki: 661nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in C6 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
BDBM26400(2,4-diamino-5,6-disubstituted pyrimidine, 14 | 9-p...)
Ki: 2.24E+3nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in C6 cells after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair