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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330459(3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]...)
Affinity DataIC50:  45.7nMAssay Description:Displacement of [3H]BRL-43694 from human 5HT3 receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Aska Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50330459(3-Amino-2-[4-(4-quinolin-2-ylpiperazin-1-yl)butyl]...)
Affinity DataEC50:  30.7nMAssay Description:Agonist activity at human cloned 5HT1A receptor expressed in CHO cells assessed as stimulation of [35S]GTPgammaS binding after 30 mins by liquid scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed