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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistamine H4 receptor(Homo sapiens (Human))
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Affinity DataKi:  2.00E+3nMAssay Description:The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H4 receptor(Homo sapiens (Human))
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Histamine H-4 Receptor Binding AssayMore data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H1 receptor(Homo sapiens (Human))
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Affinity DataIC50:  1.10E+4nMAssay Description:The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHistamine H1 receptor(Homo sapiens (Human))
Bridge Pharma

US Patent
LigandPNGBDBM181150(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Affinities of the test compounds for peripheral human histamine H-4-receptors were assessed using receptor-binding assays. The specific binding of th...More data for this Ligand-Target Pair
In DepthDetails US Patent