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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Bridge Pharma
US Patent
Ligand
BDBM181150
(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
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Affinity Data
Ki: 2.00E+3nM
Assay Description:
The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Bridge Pharma
US Patent
Ligand
BDBM181150
(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 2.00E+3nM
Assay Description:
Histamine H-4 Receptor Binding Assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Histamine H1 receptor
(Homo sapiens (Human))
Bridge Pharma
US Patent
Ligand
BDBM181150
(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.10E+4nM
Assay Description:
The specific binding of the radioactive ligand to the receptor was defined as the difference between total binding and nonspecific binding, determine...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Histamine H1 receptor
(Homo sapiens (Human))
Bridge Pharma
US Patent
Ligand
BDBM181150
(US9138431, R-NORKETOTIFEN (RNORK) | US9138431, RS-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.10E+4nM
Assay Description:
Affinities of the test compounds for peripheral human histamine H-4-receptors were assessed using receptor-binding assays. The specific binding of th...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI