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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50262479(7-Phenyl-1-(pyridazin-3-yl)-heptan-1-one | CHEMBL4...)
Affinity DataKi:  140nMpH: 9.0Assay Description:Inhibition of rat FAAH expressed in Escherichia coli at pH 9.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50262479(7-Phenyl-1-(pyridazin-3-yl)-heptan-1-one | CHEMBL4...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50262479(7-Phenyl-1-(pyridazin-3-yl)-heptan-1-one | CHEMBL4...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of TGHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50262479(7-Phenyl-1-(pyridazin-3-yl)-heptan-1-one | CHEMBL4...)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of full-length human DAGLalpha expressed in HEK293T cell membranes using para-nitrophenylbutyrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral cholesterol ester hydrolase 1(Homo sapiens (Human))
Institute For Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50262479(7-Phenyl-1-(pyridazin-3-yl)-heptan-1-one | CHEMBL4...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KIAA1363 hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed