Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50247074(7-phenyl-1-(4-(pyridin-2-yl)oxazol-2-yl)heptan-1-o...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50247074(7-phenyl-1-(4-(pyridin-2-yl)oxazol-2-yl)heptan-1-o...)
Affinity DataIC50:  30nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50247074(7-phenyl-1-(4-(pyridin-2-yl)oxazol-2-yl)heptan-1-o...)
Affinity DataIC50: <1.00E+4nMAssay Description:Inhibition of full-length human DAGLalpha expressed in HEK293T cell membranes using para-nitrophenylbutyrate by colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50247074(7-phenyl-1-(4-(pyridin-2-yl)oxazol-2-yl)heptan-1-o...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of TGH (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutral cholesterol ester hydrolase 1(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50247074(7-phenyl-1-(4-(pyridin-2-yl)oxazol-2-yl)heptan-1-o...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of KIAA1363 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed