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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Prolyl endopeptidase
(Sus scrofa)
University Of Helsinki
Curated by
ChEMBL
Ligand
BDBM50037604
(1-{(S)-2-[(S)-2-(1H-Imidazole-2-carbonyl)-pyrrolid...)
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Affinity Data
IC50: <1nM
Assay Description:
Inhibition of recombinant porcine PREP expressed in Escherichia coli using Suc-Gly-Pro-AMC as substrate preincubated for 30 mins followed by substrat...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Prolyl endopeptidase
(Sus scrofa)
University Of Helsinki
Curated by
ChEMBL
Ligand
BDBM50037604
(1-{(S)-2-[(S)-2-(1H-Imidazole-2-carbonyl)-pyrrolid...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 9nM
Assay Description:
In vitro inhibitory activity against prolyl endopeptidase (PEP)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI