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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Lethal(3)malignant brain tumor-like protein 3
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: 2.40E+3nM
Assay Description:
Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
PHD finger protein 23
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of GST-tagged PHF23 (unknown origin) using H3K4Me3 as substrate incubated for 30 mins at room temperature followed by incubation under dar...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Chromobox protein homolog 7
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of CBX7 (8 to 62) (unknown origin) expressed in Escherichia coli BL21 Rosetta DE3 using H3K9Me3 as substrate incubated for 30 mins at room...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
E3 ubiquitin-protein ligase UHRF1
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of UHRF1 tandem tudor domain (121 to 286) (unknown origin) expressed in Escherichia coli BL21 Rosetta DE3 using H3K9Me3 as substrate incub...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
TP53-binding protein 1
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of 53BP1 (1485 to 1611) (unknown origin) expressed in Escherichia coli BL21 Rosetta DE3 using H4K20Me2 as substrate incubated for 30 mins ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 5A
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+4nM
Assay Description:
Inhibition of GST-tagged Jarid1A (unknown origin) using H3K4Me3 as substrate incubated for 30 mins at room temperature followed by incubation under d...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lethal(3)malignant brain tumor-like protein 1
(Homo sapiens)
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of His-tagged L3MBTL1 (unknown origin) using H4K20Me1 as substrate incubated for 30 mins at room temperature followed by incubation under ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MBT domain-containing protein 1
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
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Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of MBTD1 (130 to 566) (unknown origin) expressed in Escherichia coli BL21 Rosetta DE3 using H4K20Me1 as substrate incubated for 30 mins at...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lethal(3)malignant brain tumor-like protein 3
(Homo sapiens (Human))
University Of North Carolina
Curated by
ChEMBL
Ligand
BDBM50496587
(CHEMBL3134138)
Copy SMILES
Copy InChI
Affinity Data
Kd: 3.80E+4nM
Assay Description:
Binding affinity to L3MBTL3 (unknown origin) by isothermal titration calorimetric analysis
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI