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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Prolyl endopeptidase FAP
(Mus musculus (Mouse))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
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Affinity Data
IC50: 64nM
Assay Description:
Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prolyl endopeptidase FAP
(Mus musculus (Mouse))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
Copy SMILES
Copy InChI
Affinity Data
IC50: 70nM
pH: 8.3 T: 2°C
Assay Description:
Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Prolyl endopeptidase
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
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Copy InChI
Affinity Data
IC50: 8.70E+3nM
Assay Description:
Inhibition of recombinant human PREP purified from Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prolyl endopeptidase
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.94E+4nM
pH: 8.3 T: 2°C
Assay Description:
Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Dipeptidyl peptidase 9
(Homo sapiens (Human))
Universiteit Antwerp
US Patent
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
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Copy InChI
Affinity Data
IC50: >5.00E+4nM
pH: 8.3 T: 2°C
Assay Description:
Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Dipeptidyl peptidase 2
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
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Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of DPP2 purified from human seminal plasma using Lys-Ala-p-nitroanilide as substrate by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dipeptidyl peptidase 4
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+5nM
Assay Description:
Inhibition of DPP4 purified from human seminal plasma using Gly-Pro-p-nitroanilide as substrate by spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Dipeptidyl peptidase 4
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+5nM
pH: 8.3 T: 2°C
Assay Description:
Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Dipeptidyl peptidase 2
(Homo sapiens (Human))
University Of Antwerp
Curated by
ChEMBL
Ligand
BDBM50009362
(CHEMBL3233838 | US9346814, Cmpd No 25 Example 29)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+5nM
pH: 8.3 T: 2°C
Assay Description:
Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI