Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 24 hits in this display
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 6.80nMAssay Description:Inhibition of SF-tagged FAP (unknown origin) expressed in Drosophila S2 cells using fluorogenic substrate by spectrometric analysisMore data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 10nMAssay Description:Inhibition of mouse recombinant FAP expressed in HEK293 cells using Ala-Pro-p-nitroanilide as substrate incubated for 15 mins prior to substrate addi...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 10nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 860nMAssay Description:Inhibition of recombinant human PREP purified from Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 860nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 860nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
BDBM233328(US9346814, Ref Cmpd No 9)
IC50: 2.40E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >4.00E+3nMAssay Description:Inhibition of SF-tagged DPP4 (unknown origin) expressed in Drosophila S2 cells using fluorogenic substrate by spectrometric analysisMore data for this Ligand-Target Pair
BDBM233328(US9346814, Ref Cmpd No 9)
IC50: 2.24E+4nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: 8.35E+4nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMAssay Description:Inhibition of DPP4 purified from human seminal plasma using Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMAssay Description:Inhibition of DPP2 purified from human seminal plasma using Lys-Ala-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM233328(US9346814, Ref Cmpd No 9)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM233328(US9346814, Ref Cmpd No 9)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM50434188(CHEMBL2385281 | US9346814, Cmpd No 2 Example 3)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
BDBM233328(US9346814, Ref Cmpd No 9)
IC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair