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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50:  3.20E+3nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProlyl endopeptidase FAP(Mus musculus (Mouse))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of recombinant mouse FAP purified from HEK293 cell supernatant using Ala-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50:  2.40E+4nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProlyl endopeptidase(Homo sapiens (Human))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of recombinant human PREP purified from Escherichia coli using Z-Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP2 purified from human seminal plasma using Lys-Ala-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of DPP4 purified from human seminal plasma using Gly-Pro-p-nitroanilide as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 2(Homo sapiens (Human))
University Of Antwerp

Curated by ChEMBL
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 9(Homo sapiens (Human))
Universiteit Antwerp

US Patent
LigandPNGBDBM50009357(CHEMBL3233575 | US9346814, Cmpd No 30 Example 35)
Affinity DataIC50: >1.00E+5nMpH: 8.3 T: 2°CAssay Description:Enzyme activities were determined kinetically in a final volume of 200 μl for 10 minutes at 37° C. by measuring the initial velocities of pNA ...More data for this Ligand-Target Pair
In DepthDetails US Patent