Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amgen

Curated by ChEMBL

LigandBDBM50459883(CHEMBL4228983)Copy SMILESCopy InChI

Affinity DataIC50:  150nMAssay Description:Inhibition of recombinant human 5-HT3A receptor expressed in HEK293 cell membranes using 5-HT as substrate in presence of [3H]GR65630More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Amgen

Curated by ChEMBL

LigandBDBM50459883(CHEMBL4228983)Copy SMILESCopy InChI

Affinity DataIC50:  1.00E+4nMAssay Description:Agonist activity at rat brain membrane alpha7 nAChRMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI