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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129073(CHEMBL64612 | [1-((3S,4S)-2-Oxo-4-phenoxy-azetidin...)
Affinity DataKi:  380nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129073(CHEMBL64612 | [1-((3S,4S)-2-Oxo-4-phenoxy-azetidin...)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129073(CHEMBL64612 | [1-((3S,4S)-2-Oxo-4-phenoxy-azetidin...)
Affinity DataKi:  3.30E+4nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129073(CHEMBL64612 | [1-((3S,4S)-2-Oxo-4-phenoxy-azetidin...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibitory activity of the compound was measured against Cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed