Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50240981(4'-piperazin-1-yl-biphenyl-4-carboxylic acid [1-(c...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity against cathepsin K using humanized rabbit enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50240981(4'-piperazin-1-yl-biphenyl-4-carboxylic acid [1-(c...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of cathepsin K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50240981(4'-piperazin-1-yl-biphenyl-4-carboxylic acid [1-(c...)
Affinity DataIC50:  614nMAssay Description:Inhibitory activity against cathepsin B from humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50240981(4'-piperazin-1-yl-biphenyl-4-carboxylic acid [1-(c...)
Affinity DataIC50:  2.27E+3nMAssay Description:Inhibitory activity against cathepsin L from humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50240981(4'-piperazin-1-yl-biphenyl-4-carboxylic acid [1-(c...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against cathepsin S from humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed