Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCathepsin S(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  1.80nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin SMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  18nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  48nMAssay Description:Compound is evaluated for inhibitory potency against CruzaineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Khepri Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50032805(CHEMBL107495 | N-[2-(3-Morpholin-4-yl-ureido)-1-na...)
Affinity DataKi:  150nMAssay Description:Compound is evaluated for inhibitory potency against cathepsin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed