Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50390593(CHEMBL2069573)
Affinity DataEC50:  930nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50390593(CHEMBL2069573)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable G-protein coupled receptor 142(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50390593(CHEMBL2069573)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human GPR142 expressed in HEK293 cells assessed as inositol phosphate accumulation using [3H]-inositol after 1 hr by scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed