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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetCaspase-3(Homo sapiens (Human))
Tianjin University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50002362(CHEMBL3233630)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human recombinant caspase-3 using Ac-LDEVD-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
Tianjin University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50002362(CHEMBL3233630)
Affinity DataIC50:  106nMAssay Description:Inhibition of recombinant human caspase-3 activity using Ac-DEVD-AMC as substrate preincubated for 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002362(CHEMBL3233630)
Affinity DataIC50:  164nMAssay Description:Inhibition of recombinant human caspase-7 activity using Ac-DEVD-AMC as substrate preincubated for 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50002362(CHEMBL3233630)
Affinity DataIC50:  909nMAssay Description:Inhibition of human recombinant caspase-7 using Ac-DEVD-AMC as substrate after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed