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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Prolyl endopeptidase
(Homo sapiens (Human))
Mcgill University
Curated by
ChEMBL
Ligand
BDBM50508977
(CHEMBL4451993)
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Affinity Data
Ki: 3.5nM
Assay Description:
Inhibition of recombinant human POP assessed as affinity constant of second step of inhibition pre-incubated for 2 hrs before addition of ZGP-pNA sub...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prolyl endopeptidase
(Homo sapiens (Human))
Mcgill University
Curated by
ChEMBL
Ligand
BDBM50508977
(CHEMBL4451993)
Copy SMILES
Copy InChI
Affinity Data
Ki: 4nM
Assay Description:
Inhibition of recombinant human POP pre-incubated for 30 mins before addition of ZGP-pNA substrate by absorbance assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prolyl endopeptidase
(Homo sapiens (Human))
Mcgill University
Curated by
ChEMBL
Ligand
BDBM50508977
(CHEMBL4451993)
Copy SMILES
Copy InChI
Affinity Data
Ki: 20nM
Assay Description:
Inhibition of recombinant human POP assessed as affinity constant of first step of the binding event pre-incubated for 2 hrs before addition of ZGP-p...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI