Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Suez Canal University

Curated by ChEMBL

LigandBDBM50143043(CHEMBL3758919)Copy SMILESCopy InChI

Affinity DataEC50:  3.02E+4nMAssay Description:Transactivation of N-terminal Gal4 DNA binding domain-linked human PPARalpha ligand binding domain after 24 hrs by luciferase reporter gene assay rel...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLMMDBPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Suez Canal University

Curated by ChEMBL

LigandBDBM50143043(CHEMBL3758919)Copy SMILESCopy InChI

Affinity DataEC50:  4.11E+3nMAssay Description:Agonist activity at human FFAR1 expressed in CHO-K1 cells assessed as calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLMMDBPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI