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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM180631(US8772323, 130)
Affinity DataEC50:  814nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM180632(US8772323, 131)
Affinity DataEC50:  7.71E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM180635(US8772323, 134)
Affinity DataEC50:  1.63E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM180634(US8772323, 133)
Affinity DataEC50:  300nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Boehringer Ingelheim International

US Patent
LigandPNGBDBM180633(US8772323, 132)
Affinity DataEC50:  4.16E+3nMpH: 7.4 T: 2°CAssay Description:MIN6 cells [Miyazaki J et al. Endocrinology. 1990 July; 127(1):126-32] were stably transfected with an expression vector for human GPR119 cDNA (Acc. ...More data for this Ligand-Target Pair
In DepthDetails US Patent