Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 7 hits in this display
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
Caspase-3(Homo sapiens (Human))Washington University
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
Caspase-6(Homo sapiens (Human))Washington University
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
Caspase-7(Homo sapiens (Human))Washington University
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
Caspase-1(Homo sapiens (Human))Washington University
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
Caspase-8(Homo sapiens (Human))Washington University
BDBM29569(acs.jmedchem.1c00409_ST.540 | isatin sulfonamide, ...)
IC50: >5.00E+4nMpH: 7.4 T: 2°CAssay Description:The caspase enzymatic activity was determined by measuring the accumulation of a fluorogenic product. All assays were prepared in 96-well format. Rec...More data for this Ligand-Target Pair