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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBromodomain-containing protein 2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(CHEMBL1363184 | LY-303511)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to BRD2 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(CHEMBL1363184 | LY-303511)
Affinity DataIC50:  9.05E+3nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to C-terminal Flag-tagged BRD4 (unknown origin) expressed in HEK293T cell nuclear extract incubated...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50210161(CHEMBL1363184 | LY-303511)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of immobilized N-LY294002 bead binding to BRD3 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed