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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Bromodomain-containing protein 2
(Homo sapiens (Human))
The University Of Sydney
Curated by
ChEMBL
Ligand
BDBM50210161
(CHEMBL1363184 | LY-303511)
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Affinity Data
IC50: 7.40E+3nM
Assay Description:
Inhibition of immobilized N-LY294002 bead binding to BRD2 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
CHEMBL
MCE
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
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Target
Bromodomain-containing protein 4
(Homo sapiens (Human))
The University Of Sydney
Curated by
ChEMBL
Ligand
BDBM50210161
(CHEMBL1363184 | LY-303511)
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Copy InChI
Affinity Data
IC50: 9.05E+3nM
Assay Description:
Inhibition of immobilized N-LY294002 bead binding to C-terminal Flag-tagged BRD4 (unknown origin) expressed in HEK293T cell nuclear extract incubated...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
MCE
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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Target
Bromodomain-containing protein 3
(Homo sapiens (Human))
The University Of Sydney
Curated by
ChEMBL
Ligand
BDBM50210161
(CHEMBL1363184 | LY-303511)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.15E+4nM
Assay Description:
Inhibition of immobilized N-LY294002 bead binding to BRD3 (unknown origin) expressed in HEK293T cell nuclear extract incubated for 1 hr by LC-MS/MS a...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
MCE
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI