Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  0.512nMAssay Description:Antagonist activity at human beta3 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  2.90nMAssay Description:Antagonist activity at human beta1 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
East China Normal University

Curated by ChEMBL
LigandPNGBDBM50462282(CHEMBL4249564)
Affinity DataEC50:  52nMAssay Description:Antagonist activity at human beta2 adrenergic receptor expressed in HEK293 cells co-expressing Galpha16 assessed as inhibition of isoproterenol-induc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed