Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetP2Y purinoceptor 12(Homo sapiens (Human))
Inspire Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371596(CHEMBL1162163)
Affinity DataIC50:  1.08E+4nMAssay Description:Antagonist activity at P2Y12 receptor assessed as inhibition of ADP-induced human platelet aggregation by washed platelet assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 6(Homo sapiens (Human))
Inspire Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371596(CHEMBL1162163)
Affinity DataEC50:  9.75E+3nMAssay Description:Agonist activity at P2Y6 receptor expressed in human 1321 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Inspire Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371596(CHEMBL1162163)
Affinity DataEC50:  2.63E+3nMAssay Description:Agonist at human recombinant P2Y1 receptor expressed in human 1321 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Inspire Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50371596(CHEMBL1162163)
Affinity DataEC50:  9.40E+3nMAssay Description:Agonist activity at P2Y2 receptor expressed in human 1321 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed