Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
BDBM50173734((2R,3R,4R,5R)-5-(5-Benzyl-[1,3,4]oxadiazol-2-yl)-2...)
Ki: 2.10E+3nMAssay Description:Inhibition constant against plasmepsin 2 of Plasmodium falciparum 10 min using 3 uM of DABCYL-Glu-Arg-Nle-Phe-Le u-Ser-Phe-Pro-EDANS as substrateMore data for this Ligand-Target Pair
BDBM50173734((2R,3R,4R,5R)-5-(5-Benzyl-[1,3,4]oxadiazol-2-yl)-2...)
Ki: >3.00E+3nMAssay Description:Inhibition constant against plasmepsin 1 of Plasmodium falciparum, 10 min using 3 uM of DABCYL-Glu-Arg-Nle-Phe-Le u-Ser-Phe-Pro-EDANS as substrateMore data for this Ligand-Target Pair
BDBM50173734((2R,3R,4R,5R)-5-(5-Benzyl-[1,3,4]oxadiazol-2-yl)-2...)