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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 16 hits in this display   

TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Tampere And Tampere University Hospital

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of human carbonic anhydrase-1 at 20 degC preincubated for 15 mins by stopped-flow CO2 hydrase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataKi:  1.16E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase IIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
University Of Tampere And Tampere University Hospital

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataKi:  2.25E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 5A, mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataKi:  3.86E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase VMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataKi:  4.26E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase IXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataKi:  4.48E+7nMAssay Description:Inhibitory activity against human Carbonic anhydrase IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 2(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant human TCPTP using pNPP as substrate measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant human PTP1B using pNPP as substrate measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataIC50:  8.05E+3nMAssay Description:In vitro inhibitory activity against recombinant human protein-tyrosine phosphatase 1B (PTP1B) using fluoreacein diphosphate (FDP) as a substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50115732(CHEMBL294467 | Sodium vanadate)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of PTP1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50:  3.02E+4nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of PP2AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50:  3.08E+4nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of PP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein phosphatase C(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50:  3.42E+4nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of CD45More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50:  3.81E+4nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of PTP-S2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50: >1.00E+6nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of LARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50094936(CHEMBL86473 | Vanadate)
Affinity DataIC50: >1.00E+6nMAssay Description:The compound was evaluated for its inhibitory activity towards Protein tyrosine phosphatase of PTP1BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed