Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetFree fatty acid receptor 1(Rattus norvegicus)
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50433707(CHEMBL2381282)
Affinity DataEC50:  77nMAssay Description:Agonist activity at GPR40 in rat INS-1 cells assessed as glucose-stimulated insulin secretionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50433707(CHEMBL2381282)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human GPR40 transfected in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50433707(CHEMBL2381282)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human GPR40 transfected in CHO cells by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed