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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM22497
(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)cyclop...)
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Affinity Data
EC50: 50nM
T: 2°C
Assay Description:
The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...
More data for this Ligand-Target Pair
Target Info
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Ligand Info
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM50475800
(CHEMBL204455)
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Affinity Data
EC50: 562nM
Assay Description:
Agonist potency at human GPR40 expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM50475785
(CHEMBL207753)
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Affinity Data
EC50: 13nM
Assay Description:
Agonist potency at human GPR40 expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM50475785
(CHEMBL207753)
Copy SMILES
Copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Agonist potency at human GPR40 expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI