Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM22497(2-(4-{[(3-phenoxyphenyl)methyl]amino}phenyl)cyclop...)
Affinity DataEC50:  50nMT: 2°CAssay Description:The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM50475800(CHEMBL204455)
Affinity DataEC50:  562nMAssay Description:Agonist potency at human GPR40 expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM50475785(CHEMBL207753)
Affinity DataEC50:  13nMAssay Description:Agonist potency at human GPR40 expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Gsk

LigandPNGBDBM50475785(CHEMBL207753)
Affinity DataEC50:  12nMAssay Description:Agonist potency at human GPR40 expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed