Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  120nMAssay Description:Agonist activity at mouse GPR120 expressed in U2OS cells assessed as induction of beta-arrestin2 recruitment after 90 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  878nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Mus musculus)
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  51nMAssay Description:Agonist activity at mouse GPR120 expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  190nMAssay Description:Agonist activity at ARMS2-PK2 -tagged human GPR120 short isoform expressed in CHOK1 cells assessed as induction of beta-arrestin2 recruitment after 9...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50208157(CHEMBL3893026 | US9708270, 30)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed