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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
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Affinity Data
EC50: 6.30E+3nM
Assay Description:
Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 220nM
Assay Description:
Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Mus musculus)
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 120nM
Assay Description:
Agonist activity at mouse GPR120 expressed in U2OS cells assessed as induction of beta-arrestin2 recruitment after 90 mins by luminescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 878nM
Assay Description:
On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 220nM
Assay Description:
Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Mus musculus)
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 51nM
Assay Description:
Agonist activity at mouse GPR120 expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 190nM
Assay Description:
Agonist activity at ARMS2-PK2 -tagged human GPR120 short isoform expressed in CHOK1 cells assessed as induction of beta-arrestin2 recruitment after 9...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50208157
(CHEMBL3893026 | US9708270, 30)
Copy SMILES
Copy InChI
Affinity Data
EC50: 6.30E+3nM
Assay Description:
Agonist activity at human GPR40 expressed in HEK293 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI