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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHistone deacetylase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50:  1.02E+4nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of full length HDAC2 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of full length HDAC3 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human full length HDAC8 expressed in Escherichia coli after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50:  3.36E+4nMAssay Description:Inhibition of full length HDAC6 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed