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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Lysine-specific demethylase 6A
(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center
Curated by
ChEMBL
Ligand
BDBM50468053
(CHEMBL4294426)
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Affinity Data
IC50: 5.50E+4nM
Assay Description:
Inhibition of KDM6A (880 to 1401 residues) (unknown origin) using H3 ( 21 to 44 residues) K27me3 as substrate preincubated for 15 min followed by sub...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
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Target
Lysine-specific demethylase 5A
(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center
Curated by
ChEMBL
Ligand
BDBM50468053
(CHEMBL4294426)
Copy SMILES
Copy InChI
Affinity Data
IC50: 8.30E+4nM
Assay Description:
Inhibition of KDM5A ARID/PhD1 domain deletion mutant (1 to 739 residues) (unknown origin) using H3 ( 1 to 24 residues) K4me3 as substrate preincubate...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
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Target
Lysine-specific demethylase 4A
(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center
Curated by
ChEMBL
Ligand
BDBM50468053
(CHEMBL4294426)
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Affinity Data
IC50: 2.90E+5nM
Assay Description:
Inhibition of KDM4A (1 to 350 residues) (unknown origin) using H3 ( 1 to 15 residues) K9me3 as substrate preincubated for 15 min followed by substrat...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Lysine-specific demethylase 5A
(Homo sapiens (Human))
The University Of Texas M.D. Anderson Cancer Center
Curated by
ChEMBL
Ligand
BDBM50468053
(CHEMBL4294426)
Copy SMILES
Copy InChI
Affinity Data
Kd: 9.00E+3nM
Assay Description:
Binding affinity to KDM5A ARID/PhD1 domain deletion mutant (1 to 588 residues) (unknown origin) by ITC assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
Article
PubMed
PDB
3D Structure (crystal)
Copy BDB DOI