Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human GPR120 short splice variant expressed in HEK293 cells assessed as increase in intracellular calcium flux incubated for 30 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human GPR40 by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  143nMAssay Description:Agonist activity at PK-tagged human GPR120 long isoform expressed in CHOK1 cells co-expressing EA-tagged beta-arrestin assessed as beta-gal enzyme co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Mus musculus)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50278673(CHEMBL4165366)
Affinity DataEC50:  77nMAssay Description:Agonist activity at mouse GPR120 by calcium flux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed