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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM22517
(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
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Affinity Data
EC50: 7.94E+3nM
T: 2°C
Assay Description:
The reporter assay for the stable hGPR40-Gal4-Elk1/5xGal4-luc+-expressing CHO cells was first carried out in the serum-free medium in the presence of...
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Target
Free fatty acid receptor 4
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM22517
(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
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Affinity Data
EC50: 5.75E+4nM
Assay Description:
Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assay
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KEGG
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
Gsk
Ligand
BDBM22517
(3-[4-(benzylamino)phenyl]propanoic acid | carboxyl...)
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Copy InChI
Affinity Data
EC50: 1.15E+3nM
Assay Description:
Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI