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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50339456
(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
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Affinity Data
Ki: 1.38E+4nM
Assay Description:
Displacement of 3-(2-Fluoro-4-((2'-methyl-4'-(2-(2-((7-nitrobenzo[c][1,2,5]-oxadiazol-4-yl)amino)ethoxy)ethoxy)-[1,1'-biphenyl]-3-yl)-methoxy)phenyl)...
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Target
Free fatty acid receptor 4
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50339456
(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
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Affinity Data
EC50: 1.17E+4nM
Assay Description:
Agonist activity at GPR120 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 5 mins by BRET assay
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KEGG
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50339456
(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
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Affinity Data
EC50: 550nM
Assay Description:
Agonist activity at FFAR1 expressed in HEK 293 cells assessed as beta-arrestin recruitment after 30 mins by BRET assay
More data for this Ligand-Target Pair
Target Info
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antibodypedia
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In Depth
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Article
PubMed
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50339456
(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
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Affinity Data
EC50: 550nM
Assay Description:
Agonist activity at human C-terminal eYFP-tagged FFA1 receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment incubated for 5 mins...
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Target Info
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antibodypedia
GoogleScholar
Ligand Info
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In Depth
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PubMed
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Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50339456
(Benzyloxyphenylpropanoic acid | CHEMBL1688452)
Copy SMILES
Copy InChI
Affinity Data
EC50: 510nM
Assay Description:
Agonist activity against human GPR40 expressed in CHO cells assessed as increase in intracellular calcium level by FLIPR assay in presence of 0.1% BS...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI