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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
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Affinity Data
EC50: 96nM
Assay Description:
Agonist activity at human FFA1 expressed in human 1321N1 cells by calcium fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 200nM
Assay Description:
Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 200nM
Assay Description:
Agonist activity at human FFA1 receptor expressed in human 1321N1 cells assessed as calcium mobilization by fluorescence spectrophotometry
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 8.51E+3nM
Assay Description:
Agonist activity at C-terminal yellow fluorescent protein-fused human FFA4 receptor transfected in HEK293 cells after 5 mins by BRET assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 1
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 200nM
Assay Description:
Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Free fatty acid receptor 4
(Homo sapiens (Human))
University Of Southern Denmark
Curated by
ChEMBL
Ligand
BDBM50275510
(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 8.51E+3nM
Assay Description:
Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI