Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50286278(CHEMBL4171403)
Affinity DataEC50:  2.36E+5nMAssay Description:Transactivation of human PPARgamma expressed in CHO cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50286278(CHEMBL4171403)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells after 24 hrs by NFAT-luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed