Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50286277(CHEMBL4168059)Copy SMILESCopy InChI

Affinity DataEC50:  2.40E+3nMAssay Description:Transactivation of human PPARgamma expressed in CHO cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL

LigandBDBM50286277(CHEMBL4168059)Copy SMILESCopy InChI

Affinity DataEC50:  38nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells after 24 hrs by NFAT-luciferase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI