Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetFree fatty acid receptor 1(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 3(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR41 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 2(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR43 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Saint Petersburg State University

Curated by ChEMBL
LigandPNGBDBM50171870(CHEMBL3805879)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human GPR120 (unknown origin) expressed in CHO cells by calcium influx assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed