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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
C-X-C chemokine receptor type 4
(Homo sapiens (Human))
Altiris Therapeutics
US Patent
Ligand
BDBM221878
(US9314468, Table 8, Compound 16)
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Affinity Data
IC50: 26nM
Assay Description:
This assay measures the change in impedance that occurs when cells are stimulated with SDF-1a. Changes in shape and cytoskeleton result in a change o...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
C-X-C chemokine receptor type 4
(Homo sapiens (Human))
Altiris Therapeutics
US Patent
Ligand
BDBM221813
(US9314468, Table 7, Compound 100 | US9314468, Tabl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 113nM
T: 2°C
Assay Description:
Functional modulation of CXCR4 was determined by calcium mobilization assay using leukemic lymphoid CEM cells, which naturally express high levels of...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
C-X-C chemokine receptor type 4
(Homo sapiens (Human))
Altiris Therapeutics
US Patent
Ligand
BDBM221813
(US9314468, Table 7, Compound 100 | US9314468, Tabl...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 135nM
T: 2°C
Assay Description:
Functional modulation of CXCR4 was determined by calcium mobilization assay using leukemic lymphoid CEM cells, which naturally express high levels of...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI