Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Altiris Therapeutics

US Patent
LigandPNGBDBM221878(US9314468, Table 8, Compound 16)
Affinity DataIC50:  26nMAssay Description:This assay measures the change in impedance that occurs when cells are stimulated with SDF-1a. Changes in shape and cytoskeleton result in a change o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Altiris Therapeutics

US Patent
LigandPNGBDBM221813(US9314468, Table 7, Compound 100 | US9314468, Tabl...)
Affinity DataIC50:  113nMT: 2°CAssay Description:Functional modulation of CXCR4 was determined by calcium mobilization assay using leukemic lymphoid CEM cells, which naturally express high levels of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Altiris Therapeutics

US Patent
LigandPNGBDBM221813(US9314468, Table 7, Compound 100 | US9314468, Tabl...)
Affinity DataIC50:  135nMT: 2°CAssay Description:Functional modulation of CXCR4 was determined by calcium mobilization assay using leukemic lymphoid CEM cells, which naturally express high levels of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent