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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50:  13nMAssay Description:Inhibition of rat liver microsome SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase 5(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50:  32nMAssay Description:Inhibition of human SCD5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50:  41nMAssay Description:Inhibition of human SCD1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA desaturase 1(Rattus norvegicus (Rat))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50:  213nMAssay Description:Inhibition of SCD1 in rat hepatocytes expressing OATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50:  7.74E+3nMAssay Description:Inhibition of SCD1 in OATP-deficient human HepG2 cells by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA 6-desaturase(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of delta-6 desaturase expressed in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA (8-3)-desaturase(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50364036(CHEMBL1950546)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of delta-5 desaturase expressed in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed