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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University of Denver and Regis University

US Patent
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataIC50:  1.40E+4nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFructose-bisphosphate aldolase(Mycobacterium tuberculosis (strain H37Rv))
The University of Denver and Regis University

US Patent
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataIC50:  1.70E+4nM Kd:  6.94E+3nMAssay Description:Enzymatic activity is measured by contacting the enzyme with a suitable substrate, such as fructose 1,6-bisphosphate, and measuring formation of a pr...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataIC50:  2.03E+5nMAssay Description:Inhibition of recombinant human QC using H-Gln-AMC hydrobromide as fluorogenic substrate incubated for 6 hrs by fluorometric microplate reader analys...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCitrate synthase, peroxisomal [1-24](Saccharomyces cerevisiae)
Nmmlsc

Curated by PubChem BioAssay
LigandPNGBDBM382(1571-30-8 | 55088_ALDRICH | 8-hydroxy-2-quinolinec...)
Affinity DataEC50:  3.00E+5nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1R03 MH086450-01 Project Title: Chemical Screen of TOR pathway GFP fusion proteins in S. ...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay