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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Cathepsin L2
(Homo sapiens (Human))
Universidade Federal De S£O Carlos
Curated by
ChEMBL
Ligand
BDBM35910
(flufenamic acid analogue, 36)
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Affinity Data
IC50: 2.10E+3nM
Assay Description:
Inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Procathepsin L
(Homo sapiens (Human))
Universidade Federal De S£O Carlos
Curated by
ChEMBL
Ligand
BDBM35910
(flufenamic acid analogue, 36)
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Affinity Data
IC50: 7.20E+3nM
Assay Description:
Inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysis
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Androgen receptor
(Homo sapiens (Human))
St. Jude Research Hospital
Ligand
BDBM35910
(flufenamic acid analogue, 36)
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Affinity Data
EC50: 3.00E+4nM
pH: 7.2 T: 2°C
Assay Description:
AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI