Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCathepsin L2(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM35910(flufenamic acid analogue, 36)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human recombinant cathepsin V expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Universidade Federal De S£O Carlos

Curated by ChEMBL
LigandPNGBDBM35910(flufenamic acid analogue, 36)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of human recombinant cathepsin L expressed in Pichia pastoris using Z-Phe-Arg-MCA as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAndrogen receptor(Homo sapiens (Human))
St. Jude Research Hospital

LigandPNGBDBM35910(flufenamic acid analogue, 36)
Affinity DataEC50:  3.00E+4nMpH: 7.2 T: 2°CAssay Description:AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed