Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
Caspase-1(Homo sapiens (Human))Procter & Gamble Pharmaceuticals
Curated by ChEMBL
BDBM50171147((S)-8-Oxo-2-phenyl-5,6,7,8-tetrahydro-1H-1,4,7a-tr...)
Caspase-8(Homo sapiens (Human))Procter & Gamble Pharmaceuticals
Curated by ChEMBL
BDBM50171147((S)-8-Oxo-2-phenyl-5,6,7,8-tetrahydro-1H-1,4,7a-tr...)
IC50: 3.05E+3nMAssay Description:Inhibitory activity towards CASP8 using fluorogenic substrates following an incubation for over 30 min at 37 degree CMore data for this Ligand-Target Pair
Caspase-3(Homo sapiens (Human))Procter & Gamble Pharmaceuticals
Curated by ChEMBL
BDBM50171147((S)-8-Oxo-2-phenyl-5,6,7,8-tetrahydro-1H-1,4,7a-tr...)
IC50: 1.00E+4nMAssay Description:Inhibitory activity towards CASP3 using fluorogenic substrates following an incubation for over 30 min at 37 degree CMore data for this Ligand-Target Pair