Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  4nMAssay Description:Inhibition of full length C-terminal FLAG-tagged human recombinant HDAC6 expressed inSf9 insect cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  290nMAssay Description:Inhibition of full length his6/FLAG-tagged human recombinant HDAC1(1 to 482 residues) expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  400nMAssay Description:Inhibition of full length C-terminal his6/FLAG-tagged human recombinant HDAC3 (1 to 2383 residues) expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  580nMAssay Description:Inhibition of full length C-terminal his6-tagged human recombinant HDAC2 (1 to 488 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of full length C-terminal his-tagged human recombinant HDAC8 expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  6.28E+3nMAssay Description:Inhibition of HDAC in human HCT-116 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of full length N-terminal GST/C-terminal his-tagged human recombinant HDAC4 (627 to 1084 residues) expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase(Homo sapiens (Human))
University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50588561(CHEMBL5193020)
Affinity DataIC50:  8.94E+3nMAssay Description:Inhibition of HDAC in human NCI-H522 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed