Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human HDAC6 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  176nMAssay Description:Inhibition of human HDAC3 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human HDAC1 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  564nMAssay Description:Inhibition of human HDAC11 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  683nMAssay Description:Inhibition of human HDAC10 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  687nMAssay Description:Inhibition of human HDAC9 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  738nMAssay Description:Inhibition of human HDAC7 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  878nMAssay Description:Inhibition of human HDAC5 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human HDAC8 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human HDAC4 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333085((R/S)-6-(6-Oxo-6,7,10,11,12,13-hexahydro-5H,9H-8,1...)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of human HDAC2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed