Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human HDAC6 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  369nMAssay Description:Inhibition of human HDAC3 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  643nMAssay Description:Inhibition of human HDAC8 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  949nMAssay Description:Inhibition of human HDAC1 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.21E+3nMAssay Description:Inhibition of human HDAC11 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of human HDAC5 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of human HDAC10 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.72E+3nMAssay Description:Inhibition of human HDAC7 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human HDAC9 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  1.93E+3nMAssay Description:Inhibition of human HDAC2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50333092((R/S)-6-(6-Oxo-6,7,9,10,11,12-hexahydro-5H-8,13-di...)
Affinity DataIC50:  2.58E+3nMAssay Description:Inhibition of human HDAC4 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed