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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetHistone deacetylase 1(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50:  9nMAssay Description:Inhibition of human recombinant full-length HDAC1 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50:  12.7nMAssay Description:Inhibition of human recombinant full-length HDAC2 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50:  23.9nMAssay Description:Inhibition of human recombinant full-length HDAC3 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50358130(CHEMBL1923808)
Affinity DataIC50:  50.2nMAssay Description:Inhibition of human recombinant full-length HDAC6 using fluorophore conjugated substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed