Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  3.10nMAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  7.90nMAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  14.5nMpH: 7.5 T: 2°CAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  18.5nMAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  43nMpH: 7.5 T: 2°CAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Illinois At Chicago

LigandPNGBDBM24349(N-[3-(1-benzyl-1H-1,2,3-triazol-4-yl)phenyl]-N'-hy...)
Affinity DataIC50:  1.99E+3nMAssay Description:The inhibitory effects of compounds on histone deacetylase (HDAC) activity were determined using a fluorescence-based assay with electrophoretic sepa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed