Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetHistone deacetylase 3(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50584251(CHEMBL5093737)
Affinity DataIC50:  13nMAssay Description:Inhibition of HDAC3 (unknown origin) incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50584251(CHEMBL5093737)
Affinity DataIC50:  30nMAssay Description:Inhibition of HDAC1 (unknown origin) incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50584251(CHEMBL5093737)
Affinity DataIC50:  54nMAssay Description:Inhibition of HDAC2 (unknown origin) incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50584251(CHEMBL5093737)
Affinity DataIC50:  71nMAssay Description:Inhibition of HDAC6 (unknown origin) incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Southeast University

Curated by ChEMBL
LigandPNGBDBM50584251(CHEMBL5093737)
Affinity DataIC50: >500nMAssay Description:Inhibition of HDAC8 (unknown origin) incubated for 30 mins by microplate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed