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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetHistone deacetylase 6(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human HDAC6 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  11nMAssay Description:Inhibition of human HDAC6 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  743nMAssay Description:Inhibition of human HDAC1 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  1.96E+3nMAssay Description:Inhibition of human HDAC2 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human HDAC11 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  5.63E+3nMAssay Description:Inhibition of human HDAC4 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  6.12E+3nMAssay Description:Inhibition of human HDAC8 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50579375(CHEMBL4858133)
Affinity DataIC50:  8.63E+3nMAssay Description:Inhibition of human HDAC10 using fluorogenic substrate incubated for 1 hrs by fluorescence plate reader assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed